Search Result "Binding kinetics"


The Role of Binding Kinetics in GPCR Drug Discovery

Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 24 Year: 2015 Page: 2504-2522
Author(s): David C. Swinney,Brad A. Haubrich,Isabelle Van Liefde,Georges Vauquelin

Can Binding Kinetics Translate to a Clinically Differentiated Drug? From Theory to Practice

Journal: Letters in Drug Design & Discovery
Volume: 3 Issue: 8 Year: 2006 Page: 569-574
Author(s): David C. Swinney

Review Article

Kinetics of Ligand Binding Through Advanced Computational Approaches: A Review

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 23 Year: 2017 Page: 2626-2641
Author(s): Alex Dickson,Pratyush Tiwary,Harish Vashisth

Drug Design for Protein Kinases and Phosphatases: Flexible-Receptor Docking, Binding Affinity and Specificity, and Drug-Binding Kinetics

Journal: Current Pharmaceutical Design
Volume: 19 Issue: 26 Year: 2013 Page: 4739-4754
Author(s): Chung F. Wong,Sneha Bairy

Review Article

Roles of Accelerated Molecular Dynamics Simulations in Predictions of Binding Kinetic Parameters

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 24 Issue: 0 Year: 2024 Page: 1-11
Author(s):

Implications of Dynamic Occupancy, Binding Kinetics, and Channel Gating Kinetics for hERG Blocker Safety Assessment and Mitigation

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 16 Year: 2016 Page: 1792-1818
Author(s): Robert A. Pearlstein,K. Andrew MacCannell,Gül Erdemli,Sarita Yeola,Gabriel Helmlinger,Qi-Ying Hu,Ramy Farid,William Egan,Steven Whitebread,Clayton Springer,Jeremy Beck,Hao-Ran Wang,Mateusz Maciejewski,Laszlo Urban,José S. Duca

Novel Experimental Design for Steady-state Processes: A Systematic Bayesian Approach for Enzymes, Drug Transport, Receptor Binding, Continuous Culture and Cell Transport Kinetics

Journal: Medicinal Chemistry
Volume: 1 Issue: 1 Year: 2005 Page: 21-29
Author(s): M. James C. Crabbe, Emma F. Murphy, Steven G. Gilmour

Enzyme Kinetics of Cytochrome P450-Mediated Reactions

Journal: Current Drug Metabolism
Volume: 2 Issue: 1 Year: 2001 Page: 17-36
Author(s): Magang Shou, Yuh Lin, Ping Lu, Cuyue Tang, Qin Mei, Dan Cui, Wei Tang, Jason S. Ngui, C. Charles Lin, Rominder Singh, Bradley K. Wong, James A. Yergey, Jiunn H. Lin, Paul G. Pearson, Thomas A. Baillie, A. David Rodrigues, Thomas H. Rushmore

Novel Functions and Binding Mechanisms of Carbohydrate-Binding Proteins Determined by Force Measurements

Journal: Current Protein & Peptide Science
Volume: 12 Issue: 8 Year: 2011 Page: 743-759
Author(s): Deborah E. Leckband

Mechanistic Evaluation of Substrate Inhibition Kinetics Observed From Aldehyde Oxidase-Catalyzed Reactions

Journal: Drug Metabolism Letters
Volume: 7 Issue: 1 Year: 2013 Page: 2-14
Author(s): Stephen W.J. Wang,Kojo Abdul-Hadi,Lawrence Cohen,Cindy Q. Xia

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